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Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism

The 18-kilodalton translocator protein (TSPO), proposed to be a key player in cholesterol transport into mitochondria, is highly expressed in steroidogenic tissues, metastatic cancer, and inflammatory and neurological diseases such as Alzheimer’s and Parkinson’s. TSPO ligands, including benzodiazepi...

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Publicado en:Science
Main Authors: Li, Fei, Liu, Jian, Zheng, Yi, Garavito, R. Michael, Ferguson-Miller, Shelagh
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5125025/
https://ncbi.nlm.nih.gov/pubmed/25635101
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.1260590
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