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Monooxorhenium(V) complexes with 222-N(2)S(2) MAMA ligands for bifunctional chelator agents: Syntheses and preliminary in vivo evaluation

INTRODUCTION: Targeted radiotherapy using the bifunctional chelate approach with (186/188)Re(V) is challenging because of the susceptibility of monooxorhenium(V)-based complexes to oxidize in vivo at high dilution. A monoamine-monoamide dithiol (MAMA)-based bifunctional chelating agent was evaluated...

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Bibliografski detalji
Izdano u:Nucl Med Biol
Glavni autori: Demoin, Dustin Wayne, Dame, Ashley N., Minard, William D., Gallazzi, Fabio, Seickman, Gary L., Rold, Tammy L., Bernskoetter, Nicole, Fassbender, Michael E., Hoffman, Timothy J., Deakyne, Carol A., Jurisson, Silvia S.
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5118109/
https://ncbi.nlm.nih.gov/pubmed/27694058
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2016.08.017
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