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Monooxorhenium(V) complexes with 222-N(2)S(2) MAMA ligands for bifunctional chelator agents: Syntheses and preliminary in vivo evaluation
INTRODUCTION: Targeted radiotherapy using the bifunctional chelate approach with (186/188)Re(V) is challenging because of the susceptibility of monooxorhenium(V)-based complexes to oxidize in vivo at high dilution. A monoamine-monoamide dithiol (MAMA)-based bifunctional chelating agent was evaluated...
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| Izdano u: | Nucl Med Biol |
|---|---|
| Glavni autori: | , , , , , , , , , , |
| Format: | Artigo |
| Jezik: | Inglês |
| Izdano: |
2016
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| Teme: | |
| Online pristup: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5118109/ https://ncbi.nlm.nih.gov/pubmed/27694058 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2016.08.017 |
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