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In Vitro Metabolic Studies of REV-ERB Agonists SR9009 and SR9011

SR9009 and SR9011 are attractive as performance-enhancing substances due to their REV-ERB agonist effects and thus circadian rhythm modulation activity. Although no pharmaceutical preparations are available yet, illicit use of SR9009 and SR9011 for doping purposes can be anticipated, especially sinc...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Geldof, Lore, Deventer, Koen, Roels, Kris, Tudela, Eva, Van Eenoo, Peter
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5085709/
https://ncbi.nlm.nih.gov/pubmed/27706103
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms17101676
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