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Optimal strategies for virtual screening of induced-fit and flexible target in the 2015 D3R Grand Challenge

Induced fit or protein flexibility can make a given structure less useful for docking and/or scoring. The 2015 Drug Design Data Resource (D3R) Grand Challenge provided a unique opportunity to prospectively test optimal strategies for virtual screening in these type of targets: heat shock protein 90...

Täydet tiedot

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Bibliografiset tiedot
Julkaisussa:J Comput Aided Mol Des
Päätekijät: Ye, Zhaofeng, Baumgartner, Matthew P., Wingert, Bentley M., Camacho, Carlos J.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2016
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC5079819/
https://ncbi.nlm.nih.gov/pubmed/27573981
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-016-9941-0
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