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Development of Solid Self-Emulsifying Formulation for Improving the Oral Bioavailability of Erlotinib
To improve the solubility and oral bioavailability of erlotinib, a poorly water-soluble anticancer drug, solid self-emulsifying drug delivery system (SEDDS) was developed using solid inert carriers such as dextran 40 and Aerosil® 200 (colloidal silica). The preliminary solubility of erlotinib in var...
Αποθηκεύτηκε σε:
| Τόπος έκδοσης: | AAPS PharmSciTech |
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| Κύριοι συγγραφείς: | , , , , , , , , |
| Μορφή: | Artigo |
| Γλώσσα: | Inglês |
| Έκδοση: |
Springer US
2015
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| Θέματα: | |
| Διαθέσιμο Online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4984901/ https://ncbi.nlm.nih.gov/pubmed/26238806 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12249-015-0370-5 |
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