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Enzymatic Macrocyclization of 1,2,3‐Triazole Peptide Mimetics

The macrocyclization of linear peptides is very often accompanied by significant improvements in their stability and biological activity. Many strategies are available for their chemical macrocyclization, however, enzyme‐mediated methods remain of great interest in terms of synthetic utility. To dat...

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Detalles Bibliográficos
Publicado en:Angew Chem Weinheim Bergstr Ger
Main Authors: Oueis, Emilia, Jaspars, Marcel, Westwood, Nicholas J., Naismith, James H.
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4924595/
https://ncbi.nlm.nih.gov/pubmed/27397939
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/ange.201601564
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