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Pro-haloacetate Nanoparticles for Efficient Cancer Therapy via Pyruvate Dehydrogenase Kinase Modulation

Anticancer agents based on haloacetic acids are developed for inhibition of pyruvate dehydrogenase kinase (PDK), an enzyme responsible for reversing the suppression of mitochondria-dependent apoptosis. Through molecular docking studies mono- and dihaloacetates are identified as potent PDK2 binders a...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Misra, Santosh K., Ye, Mao, Ostadhossein, Fatemeh, Pan, Dipanjan
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4914936/
https://ncbi.nlm.nih.gov/pubmed/27323896
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep28196
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