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Predicting Drug Extraction in the Human Gut Wall: Assessing Contributions from Drug Metabolizing Enzymes and Transporter Proteins using Preclinical Models

Intestinal metabolism can limit oral bioavailability of drugs and increase the risk of drug interactions. It is therefore important to be able to predict and quantify it in drug discovery and early development. In recent years, a plethora of models—in vivo, in situ and in vitro—have been discussed i...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Clin Pharmacokinet
Hauptverfasser: Peters, Sheila Annie, Jones, Christopher R., Ungell, Anna-Lena, Hatley, Oliver J. D.
Format: Artigo
Sprache:Inglês
Veröffentlicht: Springer International Publishing 2016
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4875961/
https://ncbi.nlm.nih.gov/pubmed/26895020
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40262-015-0351-6
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