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Efficacy of the PSD95 inhibitor Tat-NR2B9c in mice requires dose translation between species

Tat-NR2B9c, a clinical-stage stroke neuroprotectant validated in rats and primates, was recently deemed ineffective in mice. To evaluate this discrepancy, we conducted studies in mice subjected to temporary middle cerebral artery occlusion (tMCAO) for either 30 or 60 min according to the established...

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Detalhes bibliográficos
Publicado no:J Cereb Blood Flow Metab
Main Authors: Teves, Lucy M, Cui, Hong, Tymianski, Michael
Formato: Artigo
Idioma:Inglês
Publicado em: SAGE Publications 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4794097/
https://ncbi.nlm.nih.gov/pubmed/26661213
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/0271678X15612099
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