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Eliminating caspase-7 and cathepsin B cross-reactivity on fluorogenic caspase-3 substrates

11 FRET-based fluorogenic substrates were constructed using the pentapeptide template Asp-Glu-X(2)-Asp-X(1)′, and evaluated with caspase-3, caspase-7 and cathepsin B. The sequence Asp-Glu-Pro-Asp-Ser was able to selectively quantify caspase-3 activity in vitro without notable caspase-7 and cathepsin...

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Bibliografski detalji
Izdano u:Mol Biosyst
Glavni autori: Mackay, Martha, Pérez-López, Ana M., Bradley, Mark, Lilienkampf, Annamaria
Format: Artigo
Jezik:Inglês
Izdano: Royal Society of Chemistry 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4763880/
https://ncbi.nlm.nih.gov/pubmed/26726961
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5mb00730e
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