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Inhibition of G-protein-coupled Receptor Kinase 2 Prevents the Dysfunctional Cardiac Substrate Metabolism in Fatty Acid Synthase Transgenic Mice

Impairment of myocardial fatty acid substrate metabolism is characteristic of late-stage heart failure and has limited treatment options. Here, we investigated whether inhibition of G-protein-coupled receptor kinase 2 (GRK2) could counteract the disturbed substrate metabolism of late-stage heart fai...

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Pubblicato in:J Biol Chem
Autori principali: Abd Alla, Joshua, Graemer, Muriel, Fu, Xuebin, Quitterer, Ursula
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4742729/
https://ncbi.nlm.nih.gov/pubmed/26670611
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M115.702688
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