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ADMET evaluation in drug discovery: 15. Accurate prediction of rat oral acute toxicity using relevance vector machine and consensus modeling
BACKGROUND: Determination of acute toxicity, expressed as median lethal dose (LD(50)), is one of the most important steps in drug discovery pipeline. Because in vivo assays for oral acute toxicity in mammals are time-consuming and costly, there is thus an urgent need to develop in silico prediction...
Guardat en:
| Publicat a: | J Cheminform |
|---|---|
| Autors principals: | , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
Springer International Publishing
2016
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4736633/ https://ncbi.nlm.nih.gov/pubmed/26839598 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13321-016-0117-7 |
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