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CYP24 inhibition as a therapeutic target in FGF23-mediated renal phosphate wasting disorders

CYP24A1 (hereafter referred to as CYP24) enzymatic activity is pivotal in the inactivation of vitamin D metabolites. Basal renal and extrarenal CYP24 is usually low but is highly induced by its substrate 1,25-dihydroxyvitamin D. Unbalanced high and/or long-lasting CYP24 expression has been proposed...

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Detalles Bibliográficos
Publicado en:J Clin Invest
Main Authors: Bai, Xiuying, Miao, Dengshun, Xiao, Sophia, Qiu, Dinghong, St-Arnaud, René, Petkovich, Martin, Gupta, Ajay, Goltzman, David, Karaplis, Andrew C.
Formato: Artigo
Idioma:Inglês
Publicado: American Society for Clinical Investigation 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4731193/
https://ncbi.nlm.nih.gov/pubmed/26784541
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/JCI81928
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