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The ALK/ROS1 inhibitor PF-06463922 overcomes primary resistance to crizotinib in ALK-driven neuroblastoma

Neuroblastomas (NBs) harboring activating point mutations in Anaplastic Lymphoma Kinase (ALK) are differentially sensitive to the ALK inhibitor crizotinib, with certain mutations conferring intrinsic crizotinib resistance. To overcome this clinical obstacle, our goal was to identify inhibitors with...

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Publicado en:Cancer Discov
Main Authors: Infarinato, Nicole R., Park, Jin H., Krytska, Kateryna, Ryles, Hannah T., Sano, Renata, Szigety, Katherine M., Li, Yimei, Zou, Helen Y., Lee, Nathan V., Smeal, Tod, Lemmon, Mark A., Mossé, Yael P.
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4707106/
https://ncbi.nlm.nih.gov/pubmed/26554404
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/2159-8290.CD-15-1056
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