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Olaparib

Olaparib is used to treat BReast CAncer susceptibility protein (BRCA)‐associated, platinum‐sensitive ovarian cancer. Olaparib inhibits poly(ADP‐ribose) polymerase, thereby blocking the repair of single‐strand DNA breaks. This results in synthetic lethality in BRCA‐associated cancer cells, which have...

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Detalles Bibliográficos
Publicado en:Br J Clin Pharmacol
Main Authors: Goulooze, S. C., Cohen, A. F., Rissmann, R.
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4693566/
https://ncbi.nlm.nih.gov/pubmed/26344419
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.12761
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