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An engineered scorpion toxin analogue with improved Kv1.3 selectivity displays reduced conformational flexibility

The voltage-gated Kv1.3 K(+) channel plays a key role in the activation of T lymphocytes. Kv1.3 blockers selectively suppress immune responses mediated by effector memory T cells, which indicates the great potential of selective Kv1.3 inhibitors in the therapy of certain autoimmune diseases. Anuroct...

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Salvato in:
Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Bartok, Adam, Fehér, Krisztina, Bodor, Andrea, Rákosi, Kinga, Tóth, Gábor K., Kövér, Katalin E., Panyi, Gyorgy, Varga, Zoltan
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4686915/
https://ncbi.nlm.nih.gov/pubmed/26689143
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep18397
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