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Toward Improved Force-Field Accuracy through Sensitivity Analysis of Host-Guest Binding Thermodynamics

Improving the capability of atomistic computer models to predict the thermodynamics of noncovalent binding is critical for successful structure-based drug design, and the accuracy of such calculations remains limited by non-optimal force field parameters. Ideally, one would incorporate protein-ligan...

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Publicat a:J Phys Chem B
Autors principals: Yin, Jian, Fenley, Andrew T., Henriksen, Niel M., Gilson, Michael K.
Format: Artigo
Idioma:Inglês
Publicat: 2015
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4664157/
https://ncbi.nlm.nih.gov/pubmed/26181208
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jpcb.5b04262
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