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Integration of high-content screening and untargeted metabolomics for comprehensive functional annotation of natural product libraries

Traditional natural products discovery using a combination of live/dead screening followed by iterative bioassay-guided fractionation affords no information about compound structure or mode of action until late in the discovery process. This leads to high rates of rediscovery and low probabilities o...

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Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Kurita, Kenji L., Glassey, Emerson, Linington, Roger G.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4593099/
https://ncbi.nlm.nih.gov/pubmed/26371303
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1507743112
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