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Interspecies Differences in the Metabolism of Methotrexate: An Insight into the Active Site Differences between Human and Rabbit Aldehyde Oxidase

Several drug compounds have failed in clinical trials due to extensive biotransformation by aldehyde oxidase (AOX) (EC 1.2.3.1). One of the main reasons is the difficulty in scaling clearance for drugs metabolised by AOX, from preclinical species to human. Using methotrexate as a probe substrate, we...

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Bibliografski detalji
Izdano u:Biochem Pharmacol
Glavni autori: Choughule, Kanika V., Joswig-Jones, Carolyn A., Jones, Jeffrey P.
Format: Artigo
Jezik:Inglês
Izdano: 2015
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4574636/
https://ncbi.nlm.nih.gov/pubmed/26032640
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2015.05.010
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