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Simultaneous Administration of 2-Aminoethyl Diphenylborinate and Chloroquine Reverses Chloroquine Resistance in Malaria Parasites

A nearly complete reversal of chloroquine (CQ) resistance in the CQ-resistant Plasmodium falciparum K-1 strain, with a significant decrease in the mean ± standard deviation (SD) 50% inhibitory concentration (IC(50)) from 1,050 ± 95 nM to 14 ± 2 nM, was achieved in vitro by the simultaneous administr...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Main Authors: Mossaad, Ehab, Furuyama, Wakako, Enomoto, Masahiro, Kawai, Satoru, Mikoshiba, Katsuhiko, Kawazu, Shin-ichiro
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4394803/
https://ncbi.nlm.nih.gov/pubmed/25691631
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.04805-14
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