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Design, Synthesis and Evaluation of Fe-S Targeted Adenosine 5′-Phosphosulfate Reductase Inhibitors

Adenosine 5′-phosphosulfate reductase (APR) is an iron-sulfur enzyme that is vital for survival of Mycobacterium tuberculosis during dormancy and is an attractive target for the treatment of latent tuberculosis (TB) infection. The 4Fe-4S cluster is coordinated to APR by sulfur atoms of four cysteine...

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Pubblicato in:Nucleosides Nucleotides Nucleic Acids
Autori principali: Paritala, Hanumantharao, Suzuki, Yuta, Carroll, Kate S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4341950/
https://ncbi.nlm.nih.gov/pubmed/25710356
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/15257770.2014.978012
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