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Comparison of the in vitro and in vivo stability of a succinimide intermediate observed on a therapeutic IgG1 molecule

Deamidation of asparagine residues, a post-translational modification observed in proteins, is a common degradation pathway in monoclonal antibodies (mAbs). The kinetics of deamidation is influenced by primary sequence as well as secondary and tertiary folding. Analytical hydrophobic interaction chr...

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Bibliografski detalji
Glavni autori: Ouellette, David, Chumsae, Chris, Clabbers, Anca, Radziejewski, Czeslaw, Correia, Ivan
Format: Artigo
Jezik:Inglês
Izdano: Landes Bioscience 2013
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4169036/
https://ncbi.nlm.nih.gov/pubmed/23608772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4161/mabs.24458
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