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Modeling of human M1 aminopeptidases for in silico screening of potential Plasmodium falciparum alanine aminopeptidase (PfA-M1) specific inhibitors

Plasmodium falciparum alanine M1-aminopeptidase (PfA-M1) is a validated target for anti-malarial drug development. Presence of significant similarity between PfA-M1 and human M1-aminopeptidases, particularly within regions of enzyme active site leads to problem of non-specificity and off-target bind...

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Détails bibliographiques
Auteurs principaux: Sahi, Shakti, Rai, Sneha, Chaudhary, Meenakshi, Nain, Vikrant
Format: Artigo
Langue:Inglês
Publié: Biomedical Informatics 2014
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4166772/
https://ncbi.nlm.nih.gov/pubmed/25258488
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.6026/97320630010518
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