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Quantitative relationship between β-adrenergic receptor number and physiologic responses as studied with a long-lasting β-adrenergic antagonist

The aminobenzyl analog of propranolol, 1- (p-amino-α,α-dimethylphenethylamino)-3-(1-naphthoxy)-2- propanol, was synthesized and found to be a potent β-adrenergic blocking agent. The β-adrenergic receptors of cultured rat C6 glioma cells (2B clone) as assessed by [(125)I]iodohydroxybenzylpindolol bin...

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Detalhes bibliográficos
Publicado no:Proc Natl Acad Sci U S A
Principais autores: Terasaki, Wesley L., Linden, Joel, Brooker, Gary
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 1979
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC411872/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/42915/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.76.12.6401
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