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Structural Basis for Inactivation of Giardia lamblia Carbamate Kinase by Disulfiram

Carbamate kinase from Giardia lamblia is an essential enzyme for the survival of the organism. The enzyme catalyzes the final step in the arginine dihydrolase pathway converting ADP and carbamoyl phosphate to ATP and carbamate. We previously reported that disulfiram, a drug used to treat chronic alc...

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Detalhes bibliográficos
Main Authors: Galkin, Andrey, Kulakova, Liudmila, Lim, Kap, Chen, Catherine Z., Zheng, Wei, Turko, Illarion V., Herzberg, Osnat
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Biochemistry and Molecular Biology 2014
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4036171/
https://ncbi.nlm.nih.gov/pubmed/24558036
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M114.553123
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