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Targeting Oncoprotein Stability Overcomes Drug Resistance Caused by FLT3 Kinase Domain Mutations

FLT3 is the most frequently mutated kinase in acute myeloid leukemia (AML). Internal tandem duplications (ITDs) in the juxta-membrane region constitute the majority of activating FLT3 mutations. Several FLT3 kinase inhibitors were developed and tested in the clinic with significant success. However,...

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Detalhes bibliográficos
Main Authors: Yu, Chuanjiang, Kancha, Rama Krishna, Duyster, Justus
Formato: Artigo
Idioma:Inglês
Publicado em: Public Library of Science 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4029991/
https://ncbi.nlm.nih.gov/pubmed/24849514
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0097116
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