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Discovery of AZD3199, An Inhaled Ultralong Acting β(2) Receptor Agonist with Rapid Onset of Action

[Image: see text] A series of dibasic des-hydroxy β(2) receptor agonists has been prepared and evaluated for potential as inhaled ultralong acting bronchodilators. Determination of activities at the human β-adrenoreceptors demonstrated a series of highly potent and selective β(2) receptor agonists t...

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Xehetasun bibliografikoak
Egile Nagusiak: Stocks, Michael J., Alcaraz, Lilian, Bailey, Andrew, Bonnert, Roger, Cadogan, Elaine, Christie, Jadeen, Dixon, John, Connolly, Stephen, Cook, Anthony, Fisher, Adrian, Flaherty, Alice, Humphries, Alexander, Ingall, Anthony, Jordan, Stephen, Lawson, Mandy, Mullen, Alex, Nicholls, David, Paine, Stuart, Pairaudeau, Garry, Young, Alan
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Chemical Society 2014
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4027610/
https://ncbi.nlm.nih.gov/pubmed/24900851
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml4005232
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