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E3 ubiquitin ligase Cullin-5 modulates multiple molecular and cellular responses to heat shock protein 90 inhibition in human cancer cells

The molecular chaperone heat shock protein 90 (HSP90) is required for the activity and stability of its client proteins. Pharmacologic inhibition of HSP90 leads to the ubiquitin-mediated degradation of clients, particularly activated or mutant oncogenic protein kinases. Client ubiquitination occurs...

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Autors principals: Samant, Rahul S., Clarke, Paul A., Workman, Paul
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4020071/
https://ncbi.nlm.nih.gov/pubmed/24760825
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1322412111
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