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Rigid Analogues of Antimitotic Indolobenzazepinones: New Insights into Tubulin Binding via Molecular Modeling

[Image: see text] Two rigid analogues of 5-ethylindolobenzazepinone 4, a potent cytotoxic agent and inhibitor of tubulin polymerization, were prepared. The first was the indane derivative 5, in which the ethyl group is attached to the benzo moiety. The second was the pyrrolidine analogue 6, in which...

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Xehetasun bibliografikoak
Egile Nagusiak: Pons, Valérie, Beaumont, Stéphane, Tran Huu Dau, Marie Elise, Iorga, Bogdan I., Dodd, Robert H.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Chemical Society 2011
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4018049/
https://ncbi.nlm.nih.gov/pubmed/24900350
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml200024y
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