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Intramolecular arylation of benzimidazoles via Pd(II)/Cu(I) catalyzed cross-dehydrogenative coupling

Electron poor benzimidazole substrates were arylated via an intramolecular cross-dehydrogenative coupling (CDC) reaction. These CDC reactions were catalyzed by a Pd(II)/Cu(I) catalyst system, capable of producing moderate yields on a large library of substrates. The substrate scope consisted of teth...

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Библиографические подробности
Главные авторы: Pereira, Kyle C., Porter, Ashley L., DeBoef, Brenton
Формат: Artigo
Язык:Inglês
Опубликовано: 2014
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3993984/
https://ncbi.nlm.nih.gov/pubmed/24764603
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2014.01.103
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