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An Efficient, Practical, and Enantioselective Method for Synthesis of Homoallenylamides Catalyzed by an Aminoalcohol-Derived, Boron-Based Catalyst

[Image: see text] A practical catalytic method for enantioselective addition of an allene unit to aldimines is disclosed. Transformations are promoted by an in-situ-generated B-based catalyst that is derived from a simple, robust, and readily accessible (in multigram quantities) chiral aminoalcohol....

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Autori principali: Wu, Hao, Haeffner, Fredrik, Hoveyda, Amir H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2014
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3985786/
https://ncbi.nlm.nih.gov/pubmed/24588835
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja500374p
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