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Beta-endorphin-(1-27) is a naturally occurring antagonist to etorphine-induced analgesia.
The potent opioid peptide beta-endorphin is found in the brain and pituitary with two related fragments, beta-endorphin-(1-27) and beta-endorphin-(1-26). The fragments retain substantial opioid-receptor binding activity but are virtually inactive analgesically. beta-Endorphin-(1-27) inhibits beta-en...
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| Опубликовано в: : | Proc Natl Acad Sci U S A |
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| Главные авторы: | , |
| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
National Academy of Sciences
1985
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC397738/ https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/2987913/ https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.82.10.3178 |
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