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Critical Evaluation of Human Oral Bioavailability for Pharmaceutical Drugs by Using Various Cheminformatics Approaches

PURPOSE: Oral bioavailability (%F) is a key factor that determines the fate of a new drug in clinical trials. Traditionally, %F is measured using costly and time -consuming experimental tests. Developing computational models to evaluate the %F of new drugs before they are synthesized would be benefi...

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Autors principals: Kim, Marlene, Sedykh, Alexander, Chakravarti, Suman K., Saiakhov, Roustem D., Zhu, Hao
Format: Artigo
Idioma:Inglês
Publicat: 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3955412/
https://ncbi.nlm.nih.gov/pubmed/24306326
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-013-1222-1
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