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A conserved water-mediated hydrogen bond network defines bosutinib’s kinase selectivity

Kinase inhibitors are important cancer drugs, but they tend to display limited target specificity, and their target profiles are often challenging to rationalize in terms of molecular mechanism. Here we report that the clinical kinase inhibitor bosutinib recognizes its kinase targets by engaging a p...

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Autori principali: Levinson, Nicholas M., Boxer, Steven G.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3947016/
https://ncbi.nlm.nih.gov/pubmed/24292070
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.1404
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