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Antinociceptive activity of CC44, a biotinylated improgan congener

Improgan, a non-opioid, antinociceptive drug, activates descending analgesic circuits following brain administration, but the improgan receptor remains unidentified. Since biotinylation of drugs can enhance drug potency or facilitate discovery of new drug targets, a biotinylated congener of improgan...

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Autori principali: Hoerbelt, Paul, Nalwalk, Julia W., Phillips, James G., Wentland, Mark P., Shan, Zhixing, Hough, Lindsay B.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3886370/
https://ncbi.nlm.nih.gov/pubmed/23834775
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejphar.2013.06.041
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