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Identification of two calcium channel receptor sites for [3H]nitrendipine in mammalian cardiac and smooth muscle membrane.

Various Ca-channel blockers differ in cardiovascular action despite common effects at the Ca channel. Many investigators have reported only a single high-affinity receptor for binding of [3H]nitrendipine, a dihydropyridine Ca-channel blocker. Its equilibrium dissociation constant (Kd) does not match...

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Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Rogart, R B, deBruyn Kops, A, Dzau, V J
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 1986
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Accesso online:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC386736/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/2429306/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.83.19.7452
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