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Site-specific Inhibitory Mechanism for Amyloid β42 Aggregation by Catechol-type Flavonoids Targeting the Lys Residues

The aggregation of the 42-residue amyloid β-protein (Aβ42) is involved in the pathogenesis of Alzheimer disease (AD). Numerous flavonoids exhibit inhibitory activity against Aβ42 aggregation, but their mechanism remains unclear in the molecular level. Here we propose the site-specific inhibitory mec...

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Библиографические подробности
Главные авторы: Sato, Mizuho, Murakami, Kazuma, Uno, Mayumi, Nakagawa, Yu, Katayama, Sumie, Akagi, Ken-ichi, Masuda, Yuichi, Takegoshi, Kiyonori, Irie, Kazuhiro
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Biochemistry and Molecular Biology 2013
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3743493/
https://ncbi.nlm.nih.gov/pubmed/23792961
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M113.464222
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