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Synthesis and Characterization of a Novel Prostate Cancer-Targeted PI3 Kinase Inhibitor Prodrug

The phosphatidylinositol-3-kinase/Akt (PI3K/Akt) pathway is constitutively activated in a substantial proportion of prostate tumors and is considered a key mechanism supporting progression toward an androgen-independent status, for which no effective therapy is available. Therefore, PI3K inhibitors,...

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Autors principals: Baiz, Daniele, Pinder, Tanya A., Hassan, Sazzad, Karpova, Yelena, Salsbury, Freddie, Welker, Mark E., Kulik, George
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3738169/
https://ncbi.nlm.nih.gov/pubmed/22924393
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm300881a
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