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Palladium-catalyzed synthesis of N-arylated carbazoles using anilines and cyclic diaryliodonium salts

The direct synthesis of N-arylated carbazoles through a palladium-catalyzed amination of cyclic iodonium salts with anilines is described. In particular, electron-poor aniline derivatives reacted smoothly with only 5 mol % of Pd(OAc)(2) as catalyst to give the desired products in up to 71% yield. Fu...

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Autores principales: Riedmüller, Stefan, Nachtsheim, Boris J
Formato: Artigo
Lenguaje:Inglês
Publicado: Beilstein-Institut 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3701385/
https://ncbi.nlm.nih.gov/pubmed/23843915
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.9.136
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