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Iterative Refinement of a Binding Pocket Model: Active Computational Steering of Lead Optimization

[Image: see text] Computational approaches for binding affinity prediction are most frequently demonstrated through cross-validation within a series of molecules or through performance shown on a blinded test set. Here, we show how such a system performs in an iterative, temporal lead optimization e...

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Detalles Bibliográficos
Main Authors: Varela, Rocco, Walters, W. Patrick, Goldman, Brian B., Jain, Ajay N.
Formato: Artigo
Idioma:Inglês
Publicado: American Chemical Society 2012
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3640415/
https://ncbi.nlm.nih.gov/pubmed/23046104
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301210j
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