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Potent Elastase Inhibitors from Cyanobacteria: Structural Basis and Mechanisms Mediating Cytoprotective and Anti-inflammatory Effects in Bronchial Epithelial Cells

We discovered new structural diversity to a prevalent, yet medicinally underappreciated, cyanobacterial protease inhibitor scaffold and undertook comprehensive protease profiling to reveal potent and selective elastase inhibition. SAR and X-ray cocrystal structure analysis allowed a detailed assessm...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Salvador, Lilibeth A., Taori, Kanchan, Biggs, Jason S., Jakoncic, Jean, Ostrov, David A., Paul, Valerie J., Luesch, Hendrik
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2013
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3624605/
https://ncbi.nlm.nih.gov/pubmed/23350733
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm3017305
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