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Pharmacogenomics of Cytochrome P450 3A4: Recent Progress Toward the “Missing Heritability” Problem

CYP3A4 is the most important drug metabolizing enzyme in adult humans because of its prominent expression in liver and gut and because of its broad substrate specificity, which includes drugs from most therapeutic categories and many endogenous substances. Expression and function of CYP3A4 vary exte...

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Detalhes bibliográficos
Main Authors: Klein, Kathrin, Zanger, Ulrich M.
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3580761/
https://ncbi.nlm.nih.gov/pubmed/23444277
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fgene.2013.00012
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