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Facile synthesis of functionalized tetrahydroquinolines via domino Povarov reactions of arylamines, methyl propiolate and aromatic aldehydes

In the presence of p-toluenesulfonic acid as catalyst the domino reaction of arylamines, methyl propiolates and aromatic aldehydes in ethanol proceeded smoothly to give polysubstituted 1,2,3,4-tetrahydroquinolines in moderate yields. The reaction is believed to involve the Povarov reaction of in sit...

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Bibliographic Details
Main Authors: Sun, Jing, Gao, Hong, Wu, Qun, Yan, Chao-Guo
Format: Artigo
Language:Inglês
Published: Beilstein-Institut 2012
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3511020/
https://ncbi.nlm.nih.gov/pubmed/23209520
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.8.211
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