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Regulation of Inflammatory Responses in Tumor Necrosis Factor - Activated and Rheumatoid Arthritis Synovial Macrophages by Janus Kinase Inhibitors

OBJECTIVE: Inhibitors of the Janus kinases (JAKs) have been developed as anti-inflammatory and immunosuppressive agents and are currently undergoing testing in clinical trials. The JAK inhibitors CP-690,550 (tofacitinib) and INCB018424 (ruxolitinib) have demonstrated clinical efficacy in rheumatoid...

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Autores principales: Yarilina, Anna, Xu, Kai, Chan, Chunhin, Ivashkiv, Lionel B.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3510320/
https://ncbi.nlm.nih.gov/pubmed/22941906
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/art.37691
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