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Conotoxins Targeting Neuronal Voltage-Gated Sodium Channel Subtypes: Potential Analgesics?

Voltage-gated sodium channels (VGSC) are the primary mediators of electrical signal amplification and propagation in excitable cells. VGSC subtypes are diverse, with different biophysical and pharmacological properties, and varied tissue distribution. Altered VGSC expression and/or increased VGSC ac...

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Autors principals: Knapp, Oliver, McArthur, Jeffrey R., Adams, David J.
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3509706/
https://ncbi.nlm.nih.gov/pubmed/23202314
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/toxins4111236
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