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Phencyclidine (angel dust)/sigma "opiate" receptor: visualization by tritium-sensitive film.

[3H]Phencyclidine ([3H]PCP) binds specifically to an apparently single class of binding sites on slide-mounted sections of rat olfactory bulb (Kd = 46 nM; Bmax = 10.5 fmol per slice). Bound [3H]PCP can be displaced by nonradioactive PCP and a series of its analogs with relative potencies that correl...

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Publicat a:Proc Natl Acad Sci U S A
Autors principals: Quirion, R, Hammer, R P, Herkenham, M, Pert, C B
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 1981
Matèries:
Accés en línia:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC348895/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/6272322/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.78.9.5881
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