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Mutagenesis and Computer Modeling Studies of A GPCR Conserved Residue W5.43(194) in Ligand Recognition and Signal Transduction for CB2 Receptor

W5.43(194), a conserved tryptophan residue among G-protein coupled receptors (GPCRs) and cannabinoid receptors (CB), was examined in the present report for its significance in CB2 receptor ligand binding and adenylyl cyclase (AC) activity. Computer modeling postulates that this site in CB2 may be in...

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Autors principals: Zhang, Yuxun, Xie, Zhaojun, Wang, Lirong, Schreiter, Brielle, Lazo, John S., Gertsch, Jurg, Xie, Xiang-Qun
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3445262/
https://ncbi.nlm.nih.gov/pubmed/21539938
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.intimp.2011.04.013
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