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The third extracellular loop of the human calcitonin receptor-like receptor is crucial for the activation of adrenomedullin signalling

BACKGROUND AND PURPOSE: The extracellular loops (ECLs) in Family A GPCRs are important for ligand binding and receptor activation, but little is known about the function of Family B GPCR ECLs, especially ECL3. Calcitonin receptor-like receptor (CLR), a Family B GPCR, functions as a calcitonin gene-r...

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Main Authors: Kuwasako, Kenji, Hay, Debbie L, Nagata, Sayaka, Hikosaka, Tomomi, Kitamura, Kazuo, Kato, Johji
Formato: Artigo
Idioma:Inglês
Publicado: Blackwell Publishing Ltd 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3415644/
https://ncbi.nlm.nih.gov/pubmed/22142144
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2011.01803.x
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