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Designing of Protein Kinase C β-II Inhibitors against Diabetic complications: Structure Based Drug Design, Induced Fit docking and analysis of active site conformational changes

Protein Kinase C β-II (PKC β-II) is an important enzyme in the development of diabetic complications like cardiomyopathy, retinopathy, neuropathy, nephropathy and angiopathy. PKC β-II is activated in vascular tissues during diabetic vascular abnormalities. Thus, PKC β-II is considered as a potent dr...

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Detalhes bibliográficos
Main Authors: Vijayakumar, Balakrishnan, Velmurugan, Devadasan
Formato: Artigo
Idioma:Inglês
Publicado em: Biomedical Informatics 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3398787/
https://ncbi.nlm.nih.gov/pubmed/22829732
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.6026/97320630008568
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