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Quantitation of unbound sunitinib and its metabolite N-desethyl sunitinib (SU12662) in human plasma by equilibrium dialysis and liquid chromatography–tandem mass spectrometry (LC/MS/MS): application to a pharmacokinetic study

A rapid, selective, and sensitive liquid chromatography-tandem mass spectrometry method was developed and validated for the simultaneous determination of unbound sunitinib and its active metabolite N-desethyl sunitinib in plasma. Plasma and post-dialysis buffer samples were extracted using a liquid-...

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Autors principals: Rais, Rana, Zhao, Ming, He, Ping, Xu, Linping, Deeken, John F., Rudek, Michelle A.
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3382044/
https://ncbi.nlm.nih.gov/pubmed/22259028
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/bmc.2697
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